Kv11.1

1

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5

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6

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7

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13

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Chem Biol Drug Des, 2016 Jun 2 , ().

14

Ng CA et al. Tyrosine residues from the S4-S5 linker of Kv11.1 channels are critical for slow deactivation.
J. Biol. Chem., 2016 Jun 17 , ().

15

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16

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19

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20

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21

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22

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23

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24

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25

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26

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27

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28

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29

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30

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31

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32

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33

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34

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35

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36

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37

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41

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42

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46

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47

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48

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50

Lees-Miller JP et al. In response to Melgari et al. "hERG potassium channel inhibition by ivabradine requires channel gating".
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51

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52

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Heart Rhythm, 2015 Oct , 12 (2096-105).

53

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Neurosci. Lett., 2015 Nov 16 , 609 (97-102).

54

Kang Y et al. Regulation of the human ether-a-go-go-related gene (hERG) potassium channel by Nedd4 family interacting proteins (Ndfips).
Biochem. J., 2015 Nov 15 , 472 (71-82).

55

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57

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Acta Neurol. Scand., 2015 Nov , 132 (337-45).

58

Xie S et al. Hypaconitine-induced QT prolongation mediated through inhibition of KCNH2 (hERG) potassium channels in conscious dogs.
J Ethnopharmacol, 2015 May 26 , 166 (375-9).

59

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Biosens Bioelectron, 2015 May 15 , 67 (146-53).

60

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JACC Cardiovasc Imaging, 2015 May , 8 (501-10).

61

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65

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66

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67

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68

Goodchild SJ et al. Sequence of gating charge movement and pore gating in HERG activation and deactivation pathways.
Biophys. J., 2015 Mar 24 , 108 (1435-47).

69

Perissinotti LL et al. Kinetic model for NS1643 drug activation of WT and L529I variants of Kv11.1 (hERG1) potassium channel.
Biophys. J., 2015 Mar 24 , 108 (1414-24).

70

Guo J et al. NS1643 interacts around L529 of hERG to alter voltage sensor movement on the path to activation.
Biophys. J., 2015 Mar 24 , 108 (1400-13).

71

Biliczki P et al. The interaction between delayed rectifier channel alpha-subunits does not involve hetero-tetramer formation.
Naunyn Schmiedebergs Arch. Pharmacol., 2015 Mar 20 , ().

72

Lastraioli E et al. hERG1 channels drive tumour malignancy and may serve as prognostic factor in pancreatic ductal adenocarcinoma.
Br. J. Cancer, 2015 Mar 17 , 112 (1076-87).

73

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74

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Toxicol. Sci., 2015 Mar 12 , ().

75

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Zhongguo Ying Yong Sheng Li Xue Za Zhi, 2015 Mar , 31 (143-7).

76

Yang L et al. Intravenous anesthetic propofol inhibits multiple human cardiac potassium channels.
Anesthesiology, 2015 Mar , 122 (571-84).

77

Hayashi K et al. Functional Characterization of Rare Variants Implicated in Susceptibility to Lone Atrial Fibrillation.
Circ Arrhythm Electrophysiol, 2015 Jun 30 , ().

78

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79

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80

Grienke U et al. Human Ether-à-go-go Related Gene (hERG) Channel Blocking Aporphine Alkaloids from Lotus Leaves and Their Quantitative Analysis in Dietary Weight Loss Supplements.
J. Agric. Food Chem., 2015 Jun 17 , 63 (5634-9).

81

Ai Y et al. Synthesis and Biological Evaluation of Novel Olean-28,13β-lactams as Potential Antiprostate Cancer Agents.
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82

Wu W et al. The Link between Inactivation and High-Affinity Block of hERG1 Channels.
Mol. Pharmacol., 2015 Jun , 87 (1042-50).

83

Zhao X et al. Up-regulation of miR-21 and miR-23a Contributes to As2 O3 -induced hERG Channel Deficiency.
Basic Clin. Pharmacol. Toxicol., 2015 Jun , 116 (516-23).

84

Kurokawa J et al. Aromatase knockout mice reveal an impact of estrogen on drug-induced alternation of murine electrocardiography parameters.
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85

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Heart Rhythm, 2015 Jun , 12 (1306-14).

86

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Eur. J. Pharmacol., 2015 Jul 5 , 758 (97-106).

87

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Int. J. Legal Med., 2015 Jul 31 , ().

88

Zhang W et al. Kcnh2 and Kcnj8 Interactively Regulate Skin Wound Healing and Regeneration.
Wound Repair Regen, 2015 Jul 28 , ().

89

Yue Y et al. Pathogenesis of the Novel Autoimmune-Associated Long-QT Syndrome.
Circulation, 2015 Jul 28 , 132 (230-40).

90

De Mieri M et al. hERG Channel Inhibitory Daphnane Diterpenoid Orthoesters and Polycephalones A and B with Unprecedented Skeletons from Gnidia polycephala.
J. Nat. Prod., 2015 Jul 24 , 78 (1697-707).

91

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92

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93

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Int. J. Cardiol., 2015 Jul 1 , 190 (393-402).

94

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95

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96

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Mol. Pharmacol., 2015 Jul , 88 (19-28).

97

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Mol Med Rep, 2015 Jul , 12 (1233-8).

98

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Genet Test Mol Biomarkers, 2015 Jul , 19 (359-65).

99

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100

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101

Perez-Neut M et al. Stimulation of hERG1 channel activity promotes a calcium-dependent degradation of cyclin E2, but not cyclin E1, in breast cancer cells.
Oncotarget, 2015 Jan 30 , 6 (1631-9).

102

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Toxicol. Lett., 2015 Jan 22 , 232 (519-32).

103

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Bioorg. Med. Chem. Lett., 2015 Jan 1 , 25 (48-52).

104

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Physiol Rep, 2015 Jan 1 , 3 ().

105

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Phytochemistry, 2015 Jan , 109 (84-95).

106

Xiang F et al. Plectasin, first animal toxin-like fungal defensin blocking potassium channels through recognizing channel pore region.
Toxins (Basel), 2015 Jan , 7 (34-42).

107

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Fitoterapia, 2015 Jan , 100 (156-65).

108

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Eur. J. Hum. Genet., 2015 Jan , 23 (79-85).

109

Kubo T et al. Phosphatidylinositol4-phosphate 5-kinase prevents the decrease in the HERG potassium current induced by Gq protein-coupled receptor stimulation.
J. Pharmacol. Sci., 2015 Jan , 127 (127-34).

110

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Brain Res., 2015 Feb 9 , 1597 (77-85).

111

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J Biomol Screen, 2015 Feb 5 , ().

112

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J. Med. Chem., 2015 Feb 26 , 58 (1929-39).

113

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ACS Med Chem Lett, 2015 Feb 12 , 6 (210-5).

114

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Br. J. Pharmacol., 2015 Feb 12 , ().

115

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Bioorg. Med. Chem., 2015 Feb 1 , 23 (429-38).

116

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Biomed Microdevices, 2015 Feb , 17 (12).

117

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Seizure, 2015 Feb , 25 (65-7).

118

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Mol. Pharmacol., 2015 Feb , 87 (207-17).

119

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Mol. Pharmacol., 2015 Feb , 87 (338-48).

120

Gasparoli L et al. New pyrimido-indole compound CD-160130 preferentially inhibits the KV11.1B isoform and produces antileukemic effects without cardiotoxicity.
Mol. Pharmacol., 2015 Feb , 87 (183-96).

121

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ChemMedChem, 2015 Feb , 10 (276-95).

122

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123

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124

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Prog. Biophys. Mol. Biol., 2015 Dec 25 , ().

125

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126

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127

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Eur J Pharm Sci, 2015 Dec 1 , 80 (56-65).

129

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130

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131

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132

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133

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J. Med. Chem., 2015 Aug 27 , 58 (6389-409).

134

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135

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138

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139

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Clin. Pharmacol. Ther., 2015 Aug 11 , ().

141

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142

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143

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145

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146

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J. Cardiovasc. Electrophysiol., 2015 Aug , 26 (853-8).

148

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