Kv1.5

1

Wu W et al. Molecular Basis of Cardiac Delayed Rectifier Potassium Channel Function and Pharmacology.
Card Electrophysiol Clin, 2016 Jun , 8 (275-84).

2

Kojima A et al. Serum albumin attenuates the open-channel blocking effects of propofol on the human Kv1.5 channel.
Eur. J. Pharmacol., 2016 Jul 15 , 783 (117-26).

3

Subramani B et al. Generation and characterization of human cardiac resident and non-resident mesenchymal stem cell.
Cytotechnology, 2016 Jan 28 , ().

4

Lee HM et al. Blockade of Kv1.5 by paroxetine, an antidepressant drug.
Korean J. Physiol. Pharmacol., 2016 Jan , 20 (75-82).

5

Crump SM et al. Kcne4 deletion sex- and age-specifically impairs cardiac repolarization in mice.
FASEB J., 2016 Jan , 30 (360-9).

6

Ryland KE et al. Promoter Methylation Analysis Reveals That KCNA5 Ion Channel Silencing Supports Ewing Sarcoma Cell Proliferation.
Mol. Cancer Res., 2016 Jan , 14 (26-34).

7

Doczi MA et al. Developmental expression of Kv1 voltage-gated potassium channels in the avian hypothalamus.
Neurosci. Lett., 2016 Feb 1 , 616 (182-188).

8

Ou X et al. Myricetin inhibits Kv1.5 channels in HEK293 cells.
Mol Med Rep, 2016 Feb , 13 (1725-31).

9

Kajanus J et al. Isoindolinone compounds active as Kv1.5 blockers identified using a multicomponent reaction approach.
Bioorg. Med. Chem. Lett., 2016 Apr 15 , 26 (2023-9).

10

Ahmed M et al. SGK3 Sensitivity of Voltage Gated K+ Channel Kv1.5 (KCNA5).
Cell. Physiol. Biochem., 2016 , 38 (359-67).

11

Zhao Y et al. Regulation of SCN3B/scn3b by Interleukin 2 (IL-2): IL-2 modulates SCN3B/scn3b transcript expression and increases sodium current in myocardial cells.
BMC Cardiovasc Disord, 2016 , 16 (1).

12

Ohanyan V et al. Requisite Role of Kv1.5 Channels in Coronary Metabolic Dilation.
Circ. Res., 2015 Sep 11 , 117 (612-21).

13

Wang YY et al. [Effect of ERK1/2 on rat pulmonary artery smooth muscle cells Kv1.5 channel in the process of hypoxia].
Zhongguo Ying Yong Sheng Li Xue Za Zhi, 2015 Sep , 31 (418-21, 426).

14

Li P et al. E3 ligase CHIP and Hsc70 regulate Kv1.5 protein expression and function in mammalian cells.
J. Mol. Cell. Cardiol., 2015 Sep , 86 (138-46).

15

Kojima A et al. Interaction of propofol with voltage-gated human Kv1.5 channel through specific amino acids within the pore region.
Eur. J. Pharmacol., 2015 Oct 5 , 764 (622-32).

16

Asano S et al. Cecal inoculum peritonitis: An alternative model for sepsis vascular dysfunction study.
Life Sci., 2015 Nov 15 , 141 (108-18).

17

Kiper AK et al. Kv1.5 blockers preferentially inhibit TASK-1 channels: TASK-1 as a target against atrial fibrillation and obstructive sleep apnea?
Pflugers Arch., 2015 May , 467 (1081-90).

18

Fancher IS et al. Diphenyl phosphine oxide-1-sensitive K(+) channels contribute to the vascular tone and reactivity of resistance arteries from brain and skeletal muscle.
Microcirculation, 2015 May , 22 (315-25).

19

Jin SS et al. Antiarrhythmic ionic mechanism of Guanfu base A--Selective inhibition of late sodium current in isolated ventricular myocytes from guinea pigs.
Chin J Nat Med, 2015 May , 13 (361-7).

20

Lloyd J et al. Pseudosaccharin amines as potent and selective KV1.5 blockers.
Bioorg. Med. Chem. Lett., 2015 Mar 7 , ().

21

Yang L et al. Intravenous anesthetic propofol inhibits multiple human cardiac potassium channels.
Anesthesiology, 2015 Mar , 122 (571-84).

22

Turnow K et al. Interaction of DPP10a with Kv4.3 channel complex results in a sustained current component of human transient outward current Ito.
Basic Res. Cardiol., 2015 Mar , 110 (5).

23

Hayashi K et al. Functional Characterization of Rare Variants Implicated in Susceptibility to Lone Atrial Fibrillation.
Circ Arrhythm Electrophysiol, 2015 Jun 30 , ().

24

Warsi J et al. Regulation of Voltage-Gated K(+) Channel Kv1.5 by the Janus Kinase JAK3.
J. Membr. Biol., 2015 Jun 23 , ().

25

Pippucci T et al. Homozygous NOTCH3 null mutation and impaired NOTCH3 signaling in recessive early-onset arteriopathy and cavitating leukoencephalopathy.
EMBO Mol Med, 2015 Jun , 7 (848-58).

26

Yu J et al. Inhibitory effects of cortisone and hydrocortisone on human Kv1.5 channel currents.
Eur. J. Pharmacol., 2015 Jan 5 , 746 (158-66).

27

Ednie AR et al. Reduced sialylation impacts ventricular repolarization by modulating specific K+ channel isoforms distinctly.
J. Biol. Chem., 2015 Jan 30 , 290 (2769-83).

28

Chong E et al. Resveratrol, a red wine antioxidant, reduces atrial fibrillation susceptibility in the failing heart by PI3K/AKT/eNOS signaling pathway activation.
Heart Rhythm, 2015 Jan 30 , ().

29

Chapalamadugu KC et al. High level of oxygen treatment causes cardiotoxicity with arrhythmias and redox modulation.
Toxicol. Appl. Pharmacol., 2015 Jan 1 , 282 (100-7).

30

Zheng L et al. Tanshinone IIA attenuates hypoxic pulmonary hypertension via modulating KV currents.
Respir Physiol Neurobiol, 2015 Jan 1 , 205 (120-8).

31

Devalla HD et al. Atrial-like cardiomyocytes from human pluripotent stem cells are a robust preclinical model for assessing atrial-selective pharmacology.
EMBO Mol Med, 2015 Feb 19 , ().

32

Männikkö R et al. Pharmacological and electrophysiological characterisation of hERG activator AZSMO-23.
Br. J. Pharmacol., 2015 Feb 12 , ().

33

Gasparoli L et al. New pyrimido-indole compound CD-160130 preferentially inhibits the KV11.1B isoform and produces antileukemic effects without cardiotoxicity.
Mol. Pharmacol., 2015 Feb , 87 (183-96).

34

Elvira B et al. SPAK and OSR1 sensitivity of voltage-gated K+ channel Kv1.5.
J. Membr. Biol., 2015 Feb , 248 (59-66).

35

Rudakova E et al. Localization of Kv4.2 and KChIP2 in lipid rafts and modulation of outward K+ currents by membrane cholesterol content in rat left ventricular myocytes.
Pflugers Arch., 2015 Feb , 467 (299-309).

36

Ryland KE et al. Polycomb-dependent repression of the potassium channel-encoding gene KCNA5 promotes cancer cell survival under conditions of stress.
Oncogene, 2015 Aug 27 , 34 (4591-600).

37

Kidd MW et al. Intravascular pressure enhances the abundance of functional Kv1.5 channels at the surface of arterial smooth muscle cells.
Sci Signal, 2015 Aug 18 , 8 (ra83).

38

Lee JY et al. The role of K⁺ conductances in regulating membrane excitability in human gastric corpus smooth muscle.
Am. J. Physiol. Gastrointest. Liver Physiol., 2015 Apr 1 , 308 (G625-33).

39

Wang J et al. Oral administration of putrescine and proline during the suckling period improves epithelial restitution after early weaning in piglets.
J. Anim. Sci., 2015 Apr , 93 (1679-88).

40

Dai ZK et al. The Xanthine Derivative KMUP-1 Attenuates Serotonin-Induced Vasoconstriction and K⁺-Channel Inhibitory Activity via the PKC Pathway in Pulmonary Arteries.
Int. J. Biol. Sci., 2015 , 11 (633-42).

41

Lang F On the putative purpose of AMPK sensitive Kv1.5 K(+) channel regulation.
Channels (Austin), 2015 , 9 (162).

42

Yamanushi TT et al. Comparison of formaldehyde and methanol fixatives used in the detection of ion channel proteins in isolated rat ventricular myocytes by immunofluorescence labelling and confocal microscopy.
Folia Morphol. (Warsz), 2015 , 74 (258-61).

43

Ou XH et al. Remodeling of Kv1.5 channel in right atria from Han Chinese patients with atrial fibrillation.
Med. Sci. Monit., 2015 , 21 (1207-13).

44

Bartok A et al. Margatoxin is a non-selective inhibitor of human Kv1.3 K(+) channels.
Toxicon, 2014 Sep , 87 (6-16).

45

Singhal R et al. Colchicine suppresses atrial fibrillation in failing heart.
Int. J. Cardiol., 2014 Oct 20 , 176 (651-60).

46

Li B et al. Dichloroacetate prevents but not reverses the formation of neointimal lesions in a rat model of severe pulmonary arterial hypertension.
Mol Med Rep, 2014 Oct , 10 (2144-52).

47

Carrisoza-Gaytán R et al. Differential expression of the Kv1 voltage-gated potassium channel family in the rat nephron.
J. Mol. Histol., 2014 Oct , 45 (583-97).

48

Frolov RV et al. Celecoxib and ion channels: a story of unexpected discoveries.
Eur. J. Pharmacol., 2014 May 5 , 730 (61-71).

49

Fischer F et al. Isoenzyme-specific regulation of cardiac Kv1.5/Kvβ1.2 ion channel complex by protein kinase C: central role of PKCβII.
Naunyn Schmiedebergs Arch. Pharmacol., 2014 May , 387 (469-76).

50

Schumacher-Bass SM et al. Role for myosin-V motor proteins in the selective delivery of Kv channel isoforms to the membrane surface of cardiac myocytes.
Circ. Res., 2014 Mar 14 , 114 (982-92).

51

Olsson RI et al. Lactam sulfonamides as potent inhibitors of the Kv1.5 potassium ion channel.
Bioorg. Med. Chem. Lett., 2014 Mar 1 , 24 (1269-73).

52

Guo X et al. Discovery of 1-aryloxyethyl piperazine derivatives as Kv1.5 potassium channel inhibitors (part I).
Eur J Med Chem, 2014 Jun 23 , 81 (89-94).

53

Wu CT et al. Disease and region-related cardiac fibroblast potassium current variations and potential functional significance.
Cardiovasc. Res., 2014 Jun 1 , 102 (487-96).

54

Wang T et al. Muscarinic receptor activation increases hERG channel expression through phosphorylation of ubiquitin ligase Nedd4-2.
Mol. Pharmacol., 2014 Jun , 85 (877-86).

55

Johnson JA et al. Design, synthesis and evaluation of phenethylaminoheterocycles as Kv1.5 inhibitors.
Bioorg. Med. Chem. Lett., 2014 Jul 15 , 24 (3018-22).

56

Luna-Ramírez K et al. Structure, molecular modeling, and function of the novel potassium channel blocker urotoxin isolated from the venom of the Australian scorpion Urodacus yaschenkoi.
Mol. Pharmacol., 2014 Jul , 86 (28-41).

57

Iwata K et al. Deficiency of NOX1/nicotinamide adenine dinucleotide phosphate, reduced form oxidase leads to pulmonary vascular remodeling.
Arterioscler. Thromb. Vasc. Biol., 2014 Jan , 34 (110-9).

58

Wang G et al. Early onset severe pulmonary arterial hypertension with 'two-hit' digenic mutations in both BMPR2 and KCNA5 genes.
Int. J. Cardiol., 2014 Dec 20 , 177 (e167-9).

59

Vu TT et al. Soluble prokaryotic expression and purification of crotamine using an N-terminal maltose-binding protein tag.
Toxicon, 2014 Dec 15 , 92 (157-65).

60

Cidad P et al. K+ channels expression in hypertension after arterial injury, and effect of selective Kv1.3 blockade with PAP-1 on intimal hyperplasia formation.
Cardiovasc Drugs Ther, 2014 Dec , 28 (501-11).

61

Ahmed M et al. Down-regulation of K⁺ channels by human parvovirus B19 capsid protein VP1.
Biochem. Biophys. Res. Commun., 2014 Aug 8 , 450 (1396-401).

62

Schmitt N et al. Cardiac potassium channel subtypes: new roles in repolarization and arrhythmia.
Physiol. Rev., 2014 Apr , 94 (609-53).

63

Dong L et al. Potential therapeutic targets for hypoxia-induced pulmonary artery hypertension.
J Transl Med, 2014 , 12 (39).

64

Wang J et al. Effect of methamphetamine on the microglial damage: role of potassium channel Kv1.3.
PLoS ONE, 2014 , 9 (e88642).

65

Li Z et al. Exercise training reverses alterations in Kv and BKCa channel molecular expression in thoracic aorta smooth muscle cells from spontaneously hypertensive rats.
J. Vasc. Res., 2014 , 51 (447-57).

66

Nielsen JB et al. Gain-of-function mutations in potassium channel subunit KCNE2 associated with early-onset lone atrial fibrillation.
Biomark Med, 2014 , 8 (557-70).

67

Dun W et al. SAP97 and cortactin remodeling in arrhythmogenic Purkinje cells.
PLoS ONE, 2014 , 9 (e106830).

68

Odagiri F et al. Effects of candesartan on electrical remodeling in the hearts of inherited dilated cardiomyopathy model mice.
PLoS ONE, 2014 , 9 (e101838).

69

Tabarean IV Electrical remodeling of preoptic GABAergic neurons involves the Kv1.5 subunit.
PLoS ONE, 2014 , 9 (e96643).

70

Vonderlin N et al. Inhibition of cardiac Kv1.5 potassium current by the anesthetic midazolam: mode of action.
Drug Des Devel Ther, 2014 , 8 (2263-71).

71

Pousada G et al. Novel mutations in BMPR2, ACVRL1 and KCNA5 genes and hemodynamic parameters in patients with pulmonary arterial hypertension.
PLoS ONE, 2014 , 9 (e100261).

72

Baczkó I et al. Characterization of a novel multi-functional resveratrol derivative for the treatment of atrial fibrillation.
Br. J. Pharmacol., 2013 Sep 18 , ().

73

Boycott HE et al. Shear stress triggers insertion of voltage-gated potassium channels from intracellular compartments in atrial myocytes.
Proc. Natl. Acad. Sci. U.S.A., 2013 Oct 8 , 110 (E3955-E3964).

74

Olesen MS et al. Very early onset lone atrial fibrillation patients have a high prevalence of rare variants in genes previously associated with atrial fibrillation.
Heart Rhythm, 2013 Oct 18 , ().

75

Vallejo-Gracia A et al. Emerging role for the voltage-dependent K+ channel Kv1.5 in B-lymphocyte physiology: expression associated with human lymphoma malignancy.
J. Leukoc. Biol., 2013 Oct , 94 (779-89).

76

Guo X et al. Design and bio-evaluation of indole derivatives as potent Kv1.5 inhibitors.
Bioorg. Med. Chem., 2013 Nov 1 , 21 (6466-76).

77

Fedele F et al. Role of genetic polymorphisms of ion channels in the pathophysiology of coronary microvascular dysfunction and ischemic heart disease.
Basic Res. Cardiol., 2013 Nov , 108 (387).

78

Leanza L et al. Correlation between potassium channel expression and sensitivity to drug-induced cell death in tumor cell lines.
Curr. Pharm. Des., 2013 May 16 , ().

79

Christophersen IE et al. Genetic variation in KCNA5: impact on the atrial-specific potassium current IKur in patients with lone atrial fibrillation.
Eur. Heart J., 2013 May , 34 (1517-25).

80

Zhang RF et al. [Long term outcome of atrial fibrillation patients with KCNA5 and NPPA mutations post circumferential pulmonary vein ablation].
Zhonghua Xin Xue Guan Bing Za Zhi, 2013 May , 41 (387-9).

81

Finlay HJ et al. Triazolo and imidazo dihydropyrazolopyrimidine potassium channel antagonists.
Bioorg. Med. Chem. Lett., 2013 Mar 15 , 23 (1743-7).

82

Huang H et al. Diet-induced obesity causes long QT and reduces transcription of voltage-gated potassium channels.
J. Mol. Cell. Cardiol., 2013 Jun , 59 (151-8).

83

Cui Z et al. Regulation of the human ether-a-go-go-related gene (hERG) channel by Rab4 protein through neural precursor cell-expressed developmentally down-regulated protein 4-2 (Nedd4-2).
J. Biol. Chem., 2013 Jul 26 , 288 (21876-86).

84

Ravens U et al. Atrial selectivity of antiarrhythmic drugs.
J. Physiol. (Lond.), 2013 Jul 16 , ().

85

Ford J et al. Human Electrophysiological and Pharmacological Properties of XEN-D0101: A Novel Atrial Selective Kv1.5/IKur Inhibitor.
J. Cardiovasc. Pharmacol., 2013 Jan 29 , ().

86

Lang F et al. Regulation of ion channels by the serum- and glucocorticoid-inducible kinase SGK1.
FASEB J., 2013 Jan , 27 (3-12).

87

Yang Y et al. Specific Kv1.3 blockade modulates key cholesterol-metabolism-associated molecules in human macrophages exposed to ox-LDL.
J. Lipid Res., 2013 Jan , 54 (34-43).

88

Fouillade C et al. Transcriptome analysis for Notch3 target genes identifies Grip2 as a novel regulator of myogenic response in the cerebrovasculature.
Arterioscler. Thromb. Vasc. Biol., 2013 Jan , 33 (76-86).

89

Olsson RI et al. Synthesis and evaluation of diphenylphosphinic amides and diphenylphosphine oxides as inhibitors of Kv1.5.
Bioorg. Med. Chem. Lett., 2013 Feb 1 , 23 (706-10).

90

Jeong I et al. Pergolide block of the cloned Kv1.5 potassium channels.
Naunyn Schmiedebergs Arch. Pharmacol., 2013 Feb , 386 (125-33).

91

Tikhonov DB et al. Homology modeling of Kv1.5 channel block by cationic and electroneutral ligands.
Biochim. Biophys. Acta, 2013 Dec 5 , 1838 (978-987).

92

Ishii T et al. Sequestosome1/p62: a regulator of redox-sensitive voltage-activated potassium channels, arterial remodeling, inflammation, and neurite outgrowth.
Free Radic. Biol. Med., 2013 Dec , 65 (102-16).

93

Wulff H et al. Channels: Sticking to nooks and crannies.
Nat. Chem. Biol., 2013 Aug , 9 (473-4).

94

Tong M et al. Circadian expressions of cardiac ion channel genes in mouse might be associated with the central clock in the SCN but not the peripheral clock in the heart.
Biol Rhythm Res, 2013 Aug , 44 (519-530).

95

Kim SJ et al. Incretin-stimulated interaction between β-cell Kv1.5 and Kvβ2 channel proteins involves acetylation/deacetylation by CBP/SirT1.
Biochem. J., 2013 Apr 15 , 451 (227-34).

96

Gao M et al. An altered expression of genes involved in the regulation of ion channels in atrial myocytes is correlated with the risk of atrial fibrillation in patients with heart failure.
Exp Ther Med, 2013 Apr , 5 (1239-1243).

97

Atkinson AJ et al. Functional, anatomical, and molecular investigation of the cardiac conduction system and arrhythmogenic atrioventricular ring tissue in the rat heart.
J Am Heart Assoc, 2013 , 2 (e000246).

98

Mi Y et al. The role of potassium channel activation in celecoxib-induced analgesic action.
PLoS ONE, 2013 , 8 (e54797).

99

Strutz-Seebohm N et al. A Common Structural Component for β-Subunit Mediated Modulation of Slow Inactivation in Different KV Channels.
Cell. Physiol. Biochem., 2013 , 31 (968-80).

100

Zhao N et al. Potent suppression of Kv1.3 potassium channel and IL-2 secretion by diphenyl phosphine oxide-1 in human T cells.
PLoS ONE, 2013 , 8 (e64629).

101

Fujii M et al. New screening system for selective blockers of voltage-gated K(+) channels using recombinant cell lines dying upon single action potential.
J. Pharmacol. Sci., 2013 , 123 (147-58).

102

Mia S et al. Downregulation of Kv1.5 K Channels by the AMP-Activated Protein Kinase.
Cell. Physiol. Biochem., 2012 Sep 24 , 30 (1039-1050).

103

Svoboda LK et al. Redox-sensitive sulfenic acid modification regulates surface expression of the cardiovascular voltage-gated potassium channel Kv1.5.
Circ. Res., 2012 Sep 14 , 111 (842-53).

104

Lin CY et al. [Cigarette smoke exposure induced pulmonary artery pressure increase through inhibiting Kv1.5 and Kv2.1 mRNA expression in rat pulmonary artery smooth muscles].
Zhonghua Jie He He Hu Xi Za Zhi, 2012 Sep , 35 (695-9).

105

Barber AF et al. Novel activation of voltage-gated K(+) channels by sevoflurane.
J. Biol. Chem., 2012 Nov 23 , 287 (40425-32).

106

Wang T et al. Trafficking of an endogenous potassium channel in adult ventricular myocytes.
Am. J. Physiol., Cell Physiol., 2012 Nov 1 , 303 (C963-76).

107

Du YM et al. 18β-Glycyrrhetinic acid preferentially blocks late Na current generated by ΔKPQ Nav1.5 channels.
, 2012 May 21 , ().

108

Birner C et al. Differential expression of potassium channels and abnormal conduction in experimental tachycardia-induced heart failure.
Naunyn Schmiedebergs Arch. Pharmacol., 2012 May , 385 (473-80).

109

Kinoshita M et al. Sigma-1 receptor alters the kinetics of Kv1.3 voltage gated potassium channels but not the sensitivity to receptor ligands.
, 2012 Mar 6 , ().

110

Cidad P et al. Kv1.3 Channels Can Modulate Cell Proliferation During Phenotypic Switch by an Ion-Flux Independent Mechanism.
, 2012 Mar 1 , ().

111

Bielanska J et al. Differential expression of Kv1.3 and Kv1.5 voltage-dependent K+ channels in human skeletal muscle sarcomas.
Cancer Invest., 2012 Mar , 30 (203-8).

112

David M et al. Protein kinase C (PKC) activity regulates functional effects of Kvβ1.3 subunit on KV1.5 channels: identification of a cardiac Kv1.5 channelosome.
J. Biol. Chem., 2012 Jun 15 , 287 (21416-28).

113

Tipparaju SM et al. Interactions between the C-terminus of Kv1.5 and Kvβ regulate pyridine nucleotide-dependent changes in channel gating.
Pflugers Arch., 2012 Jun , 463 (799-818).

114

Gönczi M et al. Age-dependent changes in ion channel mRNA expression in canine cardiac tissues.
Gen. Physiol. Biophys., 2012 Jun , 31 (153-62).

115

Kulzer M et al. Inhibition of cardiac Kir2.1-2.3 channels by beta3 adrenoreceptor antagonist SR 59230A.
Biochem. Biophys. Res. Commun., 2012 Jul 27 , 424 (315-20).

116

Ritchie MD et al. Chromosome 4q25 Variants Are Genetic Modifiers of Rare Ion Channel Mutations Associated With Familial Atrial Fibrillation.
, 2012 Jul 10 , ().

117

Kim BS et al. Argonaute2 regulation for K+ channel-mediated human adipose tissue-derived stromal cells self-renewal and survival in nucleus.
Stem Cells Dev., 2012 Jul 1 , 21 (1736-48).

118

Dai F et al. Fluoxetine protects against big endothelin-1 induced anti-apoptosis by rescuing Kv1.5 channels in human pulmonary arterial smooth muscle cells.
Yonsei Med. J., 2012 Jul 1 , 53 (842-8).

119

Jeong I et al. Effects of dapoxetine on cloned Kv1.5 channels expressed in CHO cells.
Naunyn Schmiedebergs Arch. Pharmacol., 2012 Jul , 385 (707-16).

120

Munoz C et al. Activation of voltage gated K⁺ channel Kv1.5 by β-catenin.
Biochem. Biophys. Res. Commun., 2012 Jan 13 , 417 (692-6).

121

Li X et al. Extracellular chloride regulation of Kv2.1, contributor to the major outward Kv current in mammalian outer hair cells.
Am. J. Physiol., Cell Physiol., 2012 Jan , 302 (C296-306).

122

Jeong I et al. Carvedilol blocks the cloned cardiac Kv1.5 channels in a β-adrenergic receptor-independent manner.
Biochem. Pharmacol., 2012 Feb 15 , 83 (497-505).

123

Hald BO et al. BKCa and KV channels limit conducted vasomotor responses in rat mesenteric terminal arterioles.
Pflugers Arch., 2012 Feb , 463 (279-95).

124

Lang F et al. Serum- and glucocorticoid-inducible kinase 1 in the regulation of renal and extrarenal potassium transport.
Clin. Exp. Nephrol., 2012 Feb , 16 (73-80).

125

Suzuki S et al. Stabilization of Kv1.5 channel protein by bepridil through its action as a chemical chaperone.
Eur. J. Pharmacol., 2012 Dec 5 , 696 (28-34).

126

Schweikart K et al. The effects of jaspamide on human cardiomyocyte function and cardiac ion channel activity.
Toxicol In Vitro, 2012 Dec 20 , 27 (745-751).

127

Ishii K et al. Endocytic regulation of voltage-dependent potassium channels in the heart.
J. Pharmacol. Sci., 2012 Dec 18 , 120 (264-9).

128

Ouyang JS et al. Mitochondrial ROS-K+ channel signaling pathway regulated secretion of human pulmonary artery endothelial cells.
Free Radic. Res., 2012 Dec , 46 (1437-45).

129

Pavri BB et al. MK-0448, a specific Kv1.5 inhibitor: safety, pharmacokinetics, and pharmacodynamic electrophysiology in experimental animal models and humans.
Circ Arrhythm Electrophysiol, 2012 Dec , 5 (1193-201).

130

Qin M et al. Absence of Rgs5 prolongs cardiac repolarization and predisposes to ventricular tachyarrhythmia in mice.
J. Mol. Cell. Cardiol., 2012 Dec , 53 (880-90).

131

Liu Y et al. Effects of the natural flavone trimethylapigenin on cardiac potassium currents.
Biochem. Pharmacol., 2012 Aug 15 , 84 (498-506).

132

Dong Q et al. Hypoxia induces voltage-gated K+ (Kv) channel expression in pulmonary arterial smooth muscle cells through hypoxia-inducible factor-1 (HIF-1).
Bosn J Basic Med Sci, 2012 Aug , 12 (158-63).

133

Asano S et al. Penitrem A as a tool for understanding the role of large conductance Ca(2+)/voltage-sensitive K(+) channels in vascular function.
J. Pharmacol. Exp. Ther., 2012 Aug , 342 (453-60).

134

Felipe A et al. Targeting the voltage-dependent K(+) channels Kv1.3 and Kv1.5 as tumor biomarkers for cancer detection and prevention.
Curr. Med. Chem., 2012 , 19 (661-74).

135

Moreno C et al. Polyunsaturated Fatty acids modify the gating of kv channels.
Front Pharmacol, 2012 , 3 (163).

136

Xu XH et al. Allitridi inhibits multiple cardiac potassium channels expressed in HEK 293 cells.
PLoS ONE, 2012 , 7 (e51550).

137

Chen WL et al. Involvement of Kv1.5 protein in oxidative vascular endothelial cell injury.
PLoS ONE, 2012 , 7 (e49758).

138

Leanza L et al. Induction of apoptosis in macrophages via Kv1.3 and Kv1.5 potassium channels.
Curr. Med. Chem., 2012 , 19 (5394-404).

139

Yang XF et al. The antibody targeting the e314 Peptide of human kv1.3 pore region serves as a novel, potent and specific channel blocker.
PLoS ONE, 2012 , 7 (e36379).

140

Suzuki T et al. Multistep ion channel remodeling and lethal arrhythmia precede heart failure in a mouse model of inherited dilated cardiomyopathy.
PLoS ONE, 2012 , 7 (e35353).

141

Bossini-Castillo L et al. KCNA5 gene is not confirmed as a systemic sclerosis-related pulmonary arterial hypertension genetic susceptibility factor.
Arthritis Res. Ther., 2012 , 14 (R273).

142

Grandi E et al. Human atrial action potential and Ca2+ model: sinus rhythm and chronic atrial fibrillation.
Circ. Res., 2011 Oct 14 , 109 (1055-66).

143

Friederich P et al. The novel Kv1.5 channel blocker vernakalant for successful treatment of new-onset atrial fibrillation in a critically ill abdominal surgical patient.
Br J Anaesth, 2011 Oct , 107 (644-5).

144

Chen C et al. [Effects of puerarin on proliferation, apoptosis and Kv1.5 gene expression of pulmonary artery smooth muscle cells induced by hypoxia].
Zhonghua Lao Dong Wei Sheng Zhi Ye Bing Za Zhi, 2011 Oct , 29 (731-4).

145

Ferrer T et al. Molecular Coupling in the Human ether-a-go-go-related gene-1 (hERG1) K+ Channel Inactivation Pathway.
J. Biol. Chem., 2011 Nov 11 , 286 (39091-9).

146

Parvez B et al. The "missing" link in atrial fibrillation heritability.
J Electrocardiol, 2011 Nov , 44 (641-4).

147

Whyment AD et al. Electrophysiological, pharmacological and molecular profile of the transient outward rectifying conductance in rat sympathetic preganglionic neurons in vitro.
Neuroscience, 2011 Mar 31 , 178 (68-81).

148

Chen Y et al. The augmenter of liver regeneration protects the kidneys after orthotopic liver transplantation possibly by upregulating HIF-1α and O2-sensitive K+ channels.
Surg. Today, 2011 Mar , 41 (382-9).

149

Arvind S et al. Differential expression of a novel voltage gated potassium channel - Kv1.5 in astrocytomas and its impact on prognosis in glioblastoma.
, 2011 Jun 27 , ().

150

Hu H et al. [Effects of ethanol on action potential of rat myocardium and human Kv1.5 channel].
Sheng Li Xue Bao, 2011 Jun 25 , 63 (219-24).

151

Gurung IS et al. Deletion of the metabolic transcriptional coactivator PGC1{beta} induces cardiac arrhythmia.
, 2011 Jun 1 , ().

152

Mo J et al. Altered gene expression by low-dose arsenic exposure in humans and cultured cardiomyocytes: assessment by real-time PCR arrays.
Int J Environ Res Public Health, 2011 Jun , 8 (2090-108).

153

Goegelein H et al. Effects of the novel amiodarone-like compound SAR114646A on cardiac ion channels and ventricular arrhythmias in rats.
, 2011 Jul 16 , ().

154

Abd Allah E et al. Changes in the expression of ion channels, connexins and Ca2+ handling proteins in the sinoatrial node during postnatal development.
, 2011 Jan 28 , ().

155

Xie J et al. Dichloroacetate shifts the metabolism from glycolysis to glucose oxidation and exhibits synergistic growth inhibition with cisplatin in HeLa cells.
Int. J. Oncol., 2011 Feb , 38 (409-17).

156

Zhu S et al. Molecular diversity and functional evolution of scorpion potassium channel toxins.
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