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PubMed 18783943


Referenced in: none

Automatically associated channels: Kv11.1



Title: Overcoming hERG issues for brain-penetrating cathepsin S inhibitors: 2-cyanopyrimidines. Part 2.

Authors: Osamu Irie, Takatoshi Kosaka, Masashi Kishida, Junichi Sakaki, Keiichi Masuya, Kazuhide Konishi, Fumiaki Yokokawa, Takeru Ehara, Atsuko Iwasaki, Yuki Iwaki, Yuko Hitomi, Atsushi Toyao, Hiroki Gunji, Naoki Teno, Genji Iwasaki, Hajime Hirao, Takanori Kanazawa, Keiko Tanabe, Peter C Hiestand, Marzia Malcangio, Alyson J Fox, Stuart J Bevan, Mohammed Yaqoob, Andrew J Culshaw, Terance W Hart, Allan Hallett

Journal, date & volume: Bioorg. Med. Chem. Lett., 2008 Oct 1 , 18, 5280-4

PubMed link: http://www.ncbi.nlm.nih.gov/pubmed/18783943


Abstract