Channelpedia

PubMed 21634377


Referenced in: none

Automatically associated channels: Kv11.1 , Nav1.7



Title: Identification of a potent, state-dependent inhibitor of Nav1.7 with oral efficacy in the formalin model of persistent pain.

Authors: Howard Bregman, Loren Berry, John L Buchanan, April Chen, Bingfan Du, Elma Feric, Markus Hierl, Liyue Huang, David Immke, Brett Janosky, Danielle Johnson, Xingwen Li, Joseph Ligutti, Dong Liu, Annika Malmberg, David Matson, Jeff McDermott, Peter Miu, Hanh Nho Nguyen, Vinod F Patel, Daniel Waldon, Ben Wilenkin, Xiao Mei Zheng, Anruo Zou, Stefan I McDonough, Erin F DiMauro

Journal, date & volume: J. Med. Chem., 2011 Jul 14 , 54, 4427-45

PubMed link: http://www.ncbi.nlm.nih.gov/pubmed/21634377


Abstract