Referenced in: none

Automatically associated channels: Kv11.1

Title: Mitigating hERG Inhibition: Design of Orally Bioavailable CCR5 Antagonists as Potent Inhibitors of R5 HIV-1 Replication.

Authors: Renato Skerlj, Gary Bridger, Yuanxi Zhou, Elyse Bourque, Ernest McEachern, Sanjay Danthi, Jonathan Langille, Curtis Harwig, Duane Veale, Bryon Carpenter, Tuya Ba, Michael Bey, Ian Baird, Trevor Wilson, Markus Metz, Ron MacFarland, Renee Mosi, Veronique Bodart, Rebecca Wong, Simon Fricker, Dana Huskens, Dominique Schols

Journal, date & volume: ACS Med Chem Lett, 2012 Mar 8 , 3, 216-21

PubMed link: http://www.ncbi.nlm.nih.gov/pubmed/24900457

Abstract