Channelpedia

PubMed 18537234


Referenced in: none

Automatically associated channels: Kv11.1



Title: A novel class of cycloalkano[b]pyridines as potent and orally active opioid receptor-like 1 antagonists with minimal binding affinity to the hERG K+ channel.

Authors: Takashi Yoshizumi, Hirobumi Takahashi, Hiroshi Miyazoe, Yuichi Sugimoto, Tomohiro Tsujita, Tetsuya Kato, Hirokatsu Ito, Hiroshi Kawamoto, Mioko Hirayama, Daisuke Ichikawa, Tomoko Azuma-Kanoh, Satoshi Ozaki, Yoshihiro Shibata, Takeshi Tani, Masato Chiba, Yasuyuki Ishii, Shoki Okuda, Kiyoshi Tadano, Takahiro Fukuroda, Osamu Okamoto, Hisashi Ohta

Journal, date & volume: J. Med. Chem., 2008 Jul 10 , 51, 4021-9

PubMed link: http://www.ncbi.nlm.nih.gov/pubmed/18537234


Abstract