Channelpedia

PubMed 23886683


Referenced in: none

Automatically associated channels: Cav1.2 , Kv11.1 , Nav1.5 , TRP , TRPA , TRPA1 , TRPC , TRPC3 , TRPC6 , TRPV , TRPV1 , TRPV4



Title: The discovery of potent blockers of the canonical transient receptor channels, TRPC3 and TRPC6, based on an anilino-thiazole pharmacophore.

Authors: David G Washburn, Dennis A Holt, Jason Dodson, Jeff J McAtee, Lamont R Terrell, Linda Barton, Sharada Manns, Anna Waszkiewicz, Christina Pritchard, Dan J Gillie, Dwight M Morrow, Elizabeth A Davenport, Irina M Lozinskaya, Jeffrey Guss, Jonathan B Basilla, Lorena Kallal Negron, Michael Klein, Robert N Willette, Rusty E Fries, Timothy C Jensen, Xiaoping Xu, Christine G Schnackenberg, Joseph P Marino

Journal, date & volume: Bioorg. Med. Chem. Lett., 2013 Sep 1 , 23, 4979-84

PubMed link: http://www.ncbi.nlm.nih.gov/pubmed/23886683


Abstract