Channelpedia

PubMed 25455182


Referenced in: none

Automatically associated channels: TRP , TRPM , TRPM8



Title: Identification of a novel 2-pyridyl-benzensulfonamide derivative, RQ-00203078, as a selective and orally active TRPM8 antagonist.

Authors: Masashi Ohmi, Yuji Shishido, Tadashi Inoue, Kazuo Ando, Akiyoshi Fujiuchi, Akiko Yamada, Shuzo Watanabe, Kiyoshi Kawamura

Journal, date & volume: Bioorg. Med. Chem. Lett., 2014 Dec 1 , 24, 5364-8

PubMed link: http://www.ncbi.nlm.nih.gov/pubmed/25455182


Abstract