Channelpedia

PubMed 24884675


Referenced in: none

Automatically associated channels: TRP , TRPA , TRPA1



Title: Discovery, Optimization, and Biological Evaluation of 5-(2-(Trifluoromethyl)phenyl)indazoles as a Novel Class of Transient Receptor Potential A1 (TRPA1) Antagonists.

Authors: Lisa Rooney, Agnès Vidal, Anne-Marie D'Souza, Nick Devereux, Brian Masick, Valerie Boissel, Ryan West, Victoria Head, Rowan Stringer, Jianmin Lao, Matt J Petrus, Ardem Patapoutian, Mark Nash, Natalie Stoakley, Moh Panesar, J Martin Verkuyl, Andrew M Schumacher, H Michael Petrassi, David C Tully

Journal, date & volume: J. Med. Chem., 2014 Jun 26 , 57, 5129-40

PubMed link: http://www.ncbi.nlm.nih.gov/pubmed/24884675


Abstract